Minted: - / 5000

1148 Cartazolate
23250305c8befc7f8472f5489e6db031c0d553433c9a65a325815c7f6e06e1c3

Properties

Background

Red
Bottle

Light blue
Cap

Yellow
Syringe

Pink
Bubbles
No
Drops
Yes
Label
-

Chemistry

Formula
C15H22N4O2
Carbon
15
Polarity
Neutral

Cartazolate (SQ-65,396) is a drug of the pyrazolopyridine class. It acts as a GABA_A receptor positive allosteric modulator at the barbiturate binding site of the complex and has anxiolytic effects in animals. It is also known to act as an adenosine antagonist at the A₁ and A₂ subtypes and as a phosphodiesterase inhibitor. Cartazolate was tested in human clinical trials and was found to be efficacious for anxiety but was never marketed. It was developed by a team at E.R. Squibb and Sons in the 1970s.

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